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Home > Category > > Small Molecule Compound > ML417

ML417

Glpbio
Catalog No:GC39752-50mg CAS No.:1386162-69-1 MDLNo: Brand:Glpbio purity: 特性: Purpose:ML417 是一種選擇性的,可透過血腦屏障的 D3 多巴胺受體 (D3R) 激動劑,EC50 為 38 nM。ML417 促進 D3R 介導的 β-arrestin 易位、G 蛋白介導的信號傳導和 pERK 磷酸化,對其他 GPCR 介導的信號傳導影響最小。ML417 對毒素誘導的多巴胺能神經(jīng)元變性具有神經(jīng)保護作用。DMSO: 50 mg/mL (131.77 mM)
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