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Home > Category > > Small Molecule Compound > BI-9321 trihydrochloride

BI-9321 trihydrochloride

Glpbio
Catalog No:GC39663-100mg CAS No.:2387510-87-2 MDLNo: Brand:Glpbio purity: 特性: Purpose:BI-9321 trihydrochloride 是一種有效的,選擇性的,具有細胞活性的 NSD3-PWWP1 拮抗劑,Kd 值為 166 nM。BI-9321 對 NSD2-PWWP1 和 NSD3-PWWP2 無效。BI-9321 trihydrochloride 在 U2OS 細胞中特異性破壞 NSD3-PWWP1 與組蛋白相互作用,IC50 為 1.2 μM。DMSO: 250 mg/mL (532.13 mM)
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