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BRD5529

Glpbio
Catalog No:GC39622-100mg CAS No.:1358488-78-4 MDLNo: Brand:Glpbio purity: 特性: Purpose:BRD5529 是一種選擇性 CARD9-E3 泛素連接酶 TRIM62 蛋白-蛋白相互作用抑制劑,IC50 為 8.6 μM。BRD5529 選擇性地直接與 CARD9 結合,破壞 TRIM62 募集,抑制 TRIM62 介導的 CARD9 泛素化和激活,并在依賴 CARD9 的途徑中表現(xiàn)出細胞活性和選擇性。DMSO: 250 mg/mL (537.01 mM)
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