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Home > Category > > Small Molecule Compound > ZL0580

ZL0580

Glpbio
Catalog No:GC39576-250mg CAS No.:2377151-10-3 MDLNo: Brand:Glpbio purity: 特性: Purpose:ZL0580 是ZL0590 的結(jié)構(gòu)類似物,通過(guò)選擇性的結(jié)合到 BD1 的 BRD4 結(jié)構(gòu)域來(lái)誘導(dǎo) HIV 的表觀抑制。ZL0580通過(guò)抑制 Tat 轉(zhuǎn)錄激活和轉(zhuǎn)錄延長(zhǎng)以及在 HIV 啟動(dòng)子上誘導(dǎo)抑制染色質(zhì)結(jié)構(gòu)來(lái)誘導(dǎo) HIV 的抑制。DMSO: 250 mg/mL (469.46 mM)
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