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Home > Category > > Small Molecule Compound > PDK4-IN-1 hydrochloride

PDK4-IN-1 hydrochloride

Glpbio
Catalog No:GC39500-5mg CAS No.:2310262-11-2 MDLNo: Brand:Glpbio purity: 特性: Purpose:PDK4-IN-1 hydrochloride 是一種蒽醌衍生物,也是一種有效的,口服活性的丙酮酸脫氫酶激酶 4 (PDK4) 抑制劑,IC50 值為 84 nM。PDK4-IN-1 hydrochloride 有效抑制細胞轉化和細胞增殖并誘導細胞凋亡 (apoptosis)。PDK4-IN-1 hydrochloride 具有抗糖尿病,抗癌和抗過敏作用。DMSO: 125 mg/mL (317.36 mM)
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