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Home > Category > > Small Molecule Compound > DCLK1-IN-1

DCLK1-IN-1

Glpbio
Catalog No:GC39486-50mg CAS No.:2222635-15-4 MDLNo: Brand:Glpbio purity: 特性: Purpose:DCLK1-IN-1 是一種選擇性的、體內(nèi)相容的雙皮質(zhì)素樣激酶1 DCLK1 激酶結(jié)構(gòu)域化學(xué)探針。DCLK1-IN-1抑制 DCLK1 和 DCLK2 激酶 (結(jié)合和激酶測定 IC50 分別為: DCLK1=9.5/57.2 nM 和 DCLK2=31/103 nM)。DCLK1-IN-1 具有低毒性,可以研究 DCLK1 的生物學(xué)特性,確定其在腫瘤中的作用,如 DCLK1+ 胰腺導(dǎo)管腺癌 (PDAC)。DMSO: 35.71 mg/mL (67.69 mM)
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